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3-(1-(Dimethylamino)ethyl]phenol

3-(1-(Dimethylamino)ethyl]phenol

Fa'amatalaga Puupuu:

CAS no:105601-04-5

Mea tau vaila'au: Rivastigmine tartrate Intermediates


Fa'amatalaga Oloa

Faailoga o oloa

Fa'aoga

3-(1-(Dimethylamino)ethyl]phenol o loʻo faʻaaogaina e avea ma vaeluaga ole Rivastigmine tartrate.
Rivastigmine tartrate o rivastigmine faʻamaʻi faʻamaʻi faʻamaʻi o le Alzheimer, rivastigmine o le physostigmine derivative e Novartis mo le taimi muamua na manuia ai le atinaʻeina o le igoa tau fefaʻatauaʻiga Exelon (exelon), o se mole o loʻo i ai iina le fausaga o le carbamate, o se ituaiga amino acid o le filifili cerebral cholinesterase inhibitor, e mafai foi ona taofia. le acetylcholinesterase ma le butyrylcholinesterase, cholinergic neurons e ala i le faatuai o le faamatuu atu o le acetylcholine degradation ma le malosi faalauiloaina cholinergic neura conduction, e mafai ona faaleleia le cognitive galuega faaletonu mediated e cholinergic, faapea le faaleleia o le galuega cognitive o gasegase o le Alzheimer.Rivastigmine plasma protein fusifusia e vaivai, faigofie e ala i le toto-faiai pa, lea e maualuga le maualuga o le filifili faiʻai.E le gata e galue i luga o le cerebral cortex ma le hippocampus e sili ona faigofie ona aʻafia, ae faʻapitoa foʻi ona faʻalavelaveina le subtype iloga o le AChE i le faiʻai, e mafua ai le faʻaitiitia o le aoga o aʻafiaga itu o le cholinergic peripheral.Rivastigmine in vivo afa-ola e puupuu ma umi le umi o le gaioiga.E le pei o le tacrine, o lenei oloa i le hippocampus ma le cortex o le G1 enzyme inhibitory e malosi atu.Falema'i mo le togafitia o le tu'i leaga o le Alzheimer-type dementia, po'o le fa'ama'i Alzheimer e mafai ona masalomia ole fa'ama'i ole Alzheimer ile falema'i.


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